A blog founded by Teddy Zartler and run by Dan Erlanson for Fragment-based Drug Discovery devotees to discuss non-confidential issues regarding fragments.
Strategies for covalency:
@VividionRx recognize covalent potential on inflammasome target NLRP3, scan proteome to find cryptic site, assess promiscuity, improve selectivity, and present a chemical probe in @BrJPharmacolpracticalfragments.blogspot.…